News
- Synthese von Sulfamoylharnstoffen aus Hexafluorisopropyl-N-Fluorsulfonylcarbamat
- Photoredox-Enabled Synthesis of α-Alkylated Alkenylammonium
- Nitroxide/Nitric Acid-Promoted Oxidation of Alcohols to Aldehydes and Ketones
- Synthesis of 2-Aminothiophenes Using Piperidinium Borate
- Synthesis of Piperazin-2-ones
- Scalable Synthesis of 4-Bromo-1,2-dimethyl-1H-imidazole
- Primary Benzylic Amines via Copper-Catalyzed Benzylic C(sp3)–H Carbamation
- Novel tert-Butylation of Carboxylic Acids and Alcohols
- Synthesis of Squaric Acid Monoamides as Building Blocks for Drug Discovery
- Synthesis of Glucuronic Acid-Containing Fragments of a Heparin Sulfate Mimetic
- Synthesis of Benzo[b]azepines with a Fluorinated Side Chain
- Mechanochemical Silver-Catalyzed Ring-Opening Fluorination of Cyclobutanols
- Synthesis of Acidiphilamides A–C
- Total Synthesis of Bio-orthogonally Functionalized Securinega Alkaloids
- Visible-Light-Mediated Regioselective Chlorosulfonylation of Acrylamides
- Enantioselective Synthesis of Antispasmodic Drug (R)-Tiagabine
- Synthesis of Trisubstituted Furans from Homopropargylic Alcohols
- Photochemical Flow Synthesis of Pyrazolines from Tetrazoles
- Gold-Catalyzed Stereoselective Synthesis of Polysubstituted Indanes
- Organocatalytic Synthesis of γ-Amino Acid Precursors
- Oxidation of α-CF3 and Other Secondary Alcohols to Ketones Using a Nitroxide Catalyst
- Regioselective Synthesis of 5-Substituted Pyrazoles
- Synthesis of the Proposed Structure of Cryptoconcatone H
- One-Step and Gram-Scale Synthesis of Caffeine-d9
- Bromothiolation of Internal Alkynes
- Photooxidation of Toluene Derivatives into Carboxylic Acids
- One-Pot Synthesis of Diaryl Sulfonamides via Metal Catalysis
- Gram-Scale Synthesis of Substituted Triarylmethanes
- Synthesis of [10]Cycloparaphenylenes and their Binding to C60
- Improved Scalable Synthesis of the (S,S)-DACH-Ph Trost Ligand
- Rh(II)-Catalyzed N–H Amination of Aliphatic Amines and α-Amino Acids
- Novel Nickel-Catalyzed Synthesis of (Trifluoromethyl)quinolines
- Synthesis of Quaternary α-Fluoronitriles from Monofluorolkenes
- Stereoselective Synthesis of (–)-Heliannuol E
- General Entry to Pyrazolo[3,4-b]pyridine-3-carboxamides
- Seven-Step Synthesis of (±)-epi-Costunolide
- Total Synthesis of a Microbiologically Important Pentasaccharide
- Synthesis of the Selective Serotonin 2A Receptor Agonist 25CN-NBOH
- Synthesis of Ar-SF4Cl and Ar-SF5 Compounds from Arylphosphorothiolates
- Entry to N-Protected Serine/Threonine-Derived Weinreb Amides
- Oxa-(4+4)-Cycloaddition Entry to Oxazocine Scaffolds
- Concise Total Synthesis of (+)-Aphanorphine
- Synthesis of Allyl Aryl Sulfones from Morita–Baylis–Hillman Adducts and Thiosulfonates
- Fe(III)-Catalyzed Synthesis of 1-Chalcogenylated Naphthalene Derivatives
- Catalytic Synthesis of Olivetol and Derivatives
- Nickel-Catalyzed Synthesis of Benzofuran Derivatives
- Synthesis of Fluorenone-Fused Coumarins
- Stereoselective Synthesis of the Cotylenin A Aglycone Carbon Skeleton
- Novel Entry to Fluorinated Cyclopropanes
- Ni-H-Catalyzed Isomerization-Induced Cleavage of Allyl Ethers
- Continuous Photochemical Benzyne-Forming Process
- Copper-Catalyzed Ring Expansion of Vinyl Aziridines
- Synthesis of Constrained Benzoxazepines and Imidazopyrazines
- Synthesis of N-Aryl-1,2,3,4-tetrahydroisoquinolines
- A Molecular Stereostructure Descriptor for Asymmetric Catalysis
- A Catalytic One-Pot Synthesis of Indolyl Cyclobutanones
- Vitamin B12-Photo-Catalyzed Dicarbofunctionalization of Bromoalkenes
- Scalable Synthesis of Thiazole Peptide Macrocycles
- Synthesis of Optically Active Maresin 2
- Decarbonylative Alkynylation of Acyl Fluorides
- First Total Synthesis of the Alkaloid Clausenalansine A
- Synthesis of 4,5-Diaryl-2H-1,2,3-triazoles
- Diastereoselective Total Synthesis of (±)-Parvistemonine A
- Synthesis of Thienyl Thioethers and Thieno[3,2-b]thiophenes
- Synthesis of an Azabicyclo[3.1.0]hexanone Drug Candidate
- Redox-Neutral C1-Alkynylation of Tetrahydroisoquinolines
- Synthesis of Secondary Alcohols from Alkynes in Water
- Synthesis of Fused-ring Heptacyclic Pyrrolidines
- Peptide Synthesis with α,α-Difluoro-β-Lactams
- Synthesis of 13,19,20-Trihydroxy Docosahexaenoic Acid Stereoisomers
- Propargylation of Diaryl Azo Compounds
- Total Synthesis of Phyllanemblinin B
- Synthesis and Structure of 1-Substituted Semithioglycolurils
- Copper-Catalyzed Stereoselective Synthesis of 2-Deoxygalactosides
- Synthesis of Alkyl-methyl/ethyl Derivatives from N-(Acyloxyalkyl)phthalimides
- Synthesis of N-Substituted Ureas from Primary Amides
- Regioselective Synthesis of 3,5-Disubstituted Pyrazoles
- Synthesis of Hybrid Chromone/Coumarin 3-Halo-1H-indenes
- Annulation Approach to Tetrahydro-1,2,4-triazinecarboxylate Esters
- Scalable Synthesis of Sphingomyelins
- Synthesis of Polycyclic Indolines
- Diels–Alder Based Approach to Prenyleudesmane Diterpenoids
- Total Synthesis of Glycosyl Flavonoids
- Total Synthesis of Asparenydiol
- Synthesis of the Enantiomers of Thioridazine
- Novel Synthesis of Benzoxazoles and Benzimidazoles
- A Study of Samarium(II)–Water Allylic Benzoate Reductions
- Formal Synthesis of Pseudolaric Acid B
- Metal-Free Synthesis of Hindered 3-Azoindoles
- Multigram Deoxofluorination of β-Keto Esters with Sulfur Tetrafluoride
- A Radical-Chemistry Approach to 2-Arylquinolines
- Novel 2-Substituted Analogues of (–)-Pentenomycin I
- Detailed Comparison of Ni vs. Pd in Cross-Coupling Catalysis
- Synthesis of Sulfonylisoureas via Sulfo-Click Reactions
- Selenium Tetrachloride Catalyzed Iodination of (Hetero)Arenes
- Pd-Catalyzed Synthesis of N-Allyloxypyrrolidinediones
- A Novel Approach to Diarylated Esters and Phosphonates
- One-Pot Access to 2-Aryl-3-(arylmethyl)chromones
- Benzoazepinoindoles – A New Class of Heterocycles
- Metal-Free Hydroamination of Alkynes
- 1,2,4,5-Tetrazine Derivatives from Arylsulfonylhydrazones
- Mono- and Dihalogenation of 2-Aminopyrazine
- Novel Approach to Antihistamine-type Scaffolds
- Poster Prize awarded at ISySyCat 2019
- An Improved Synthesis of 2,5-Disubstituted Tetrazoles
- Total Synthesis of Shensongine A
- Synthesis of Novel Imidazothiadiazoles
- Cu(II)-Catalyzed Beckmann Rearrangement of Ketones
- Allylic C–H Alkynylation via Copper Photocatalysis
- Synthesis of Dumbbell-like Amine-Functionalized Bis-C60 Fullerene
- It was not tricyanomethane, after all…
- Total Syntheses of (+)-Alexine and Related Alkaloids
- Poster Prize awarded at Bioheterocycles 2019
- Photoredox Fischer Indole Synthesis
- Synthesis of Resolvins and Derivatives
- Poster Prize awarded at Twente / Mainz Symposium
- First Total Synthesis of Artekeiskeanol A, C and Altissimacoumarin D
- Iodoglycosylation and Iodocarboxylation of Glycals
- Gold(III)-Catalyzed Synthesis of N,N-Aryl,Benzyl-amines in Water
- Synthesis of Fatty Acid Intermediates via Hudrlik–Peterson Reaction
- Recyclable Graphene Oxide Nanosheet Supported Catalyst
- A Stereoselective Synthesis of the ACE Inhibitor Trandolapril
- New Entry to 3-Arylglutaconic Acid Derivatives
- Electrochemical C(sp³)–H Fluorination
- Asymmetric Synthesis of α-Hydrazino Ketones
- Synthesis of (–)-Boschnialactone and γ-Lycorane
- Synthesis of the ABC-Ring System of Various Alkaloids
- Regioselective Halogenation of Coumarins
- Synthesis of 4-(Arylmethyl)proline Derivatives
- Efficient Synthesis of a 5α-Reductase Inhibitor
- Epoxidation of a Cyclic Allyl-Amine by a Bifunctional Peracid
- Radiochemical Synthesis of 2-[18F]Fluorophenylalanine
- Asymmetric Mannich-Type Reaction of an α-Trifluoromethyl Amide
- Chemoselective Aerobic Oxidation of Benzylic Alcohols
- One-Pot Reductive Conversion of Aldehydes into Acetic Esters
- Visible-Light-Induced Adamantylation of Azoles
- Synthesis of Protected Stereodefined 5-Aminomethylprolines
- Synthesis of Thiophene-Fused 1,10-Phenanthrolines
- Synthesis of 8-Oxabicyclo[3.2.1]octanes
- Asymmetric Synthesis of Netarsudil
- Borylated Cyclohexenes via Suzuki–Miyaura/Diels–Alder Cascade
- Synthesis of 1-Alkylisoquinolines via Radical Cyclization
- Biphenyls via Cross-Coupling of Arenediazonium Salts
- Synthesis of Anthraquinones via Pd-Catalyzed Acylation
- Synthesis and Applications of 4-Chloro-2-(trichloromethyl)pyrimidines
- Catalyzed Conversion of Aldehydes into Nitriles
- Synthesis of Aryl/Heteroaryl Amides via Nitriles Hydration
- Stereospecific Amination of Alkylboronic Esters
- Metathesis Reactions for Accessing β-Amino Acid Derivatives
- Selective Preparation of C2v-Symmetric Hexaphenylbenzenes
- Stereoselective Oxidation of Titanium(IV) Enolates with Oxygen
- Ring-Closing Metathesis Entry to Dienamide Heterocycles
- New Dipeptide Organocatalysts for Aldol Reactions
- A Biomimetic Synthesis of des-Hydroxy Paecilospirone
- Monitoring Solid-Phase Reactions with Thin-Layer Chromatography
- Multi-Component Synthesis of N-Unsubstituted 1,2,3-Triazoles
- Organocatalytic Enantioselective Synthesis of 1,3-Disubstituted Allenols
- Improved Synthesis of Guanine Quadruplex Ligand Phen-DC3
- C–H Alkylation of Heteroarenes with Alkyl Bromides
- Synthesis of Nepetoidin B
- Synthesis of 2-Azabicyclo[n.2.0]alkane-Derived Building Blocks
- Novel Approach to Organo-Phosphinates and Phosphonates
- Conceptually New Approach to Ellipticine and the Oxoaporphine Core
- Difluoro(phenylsulfanyl)methane as a Formylating Agent
- Synthesis of a Gallium Complexing Agent used in PET Tracers
- Increasing Tetrazine Reactivity in the IEDDA Reaction
- Multicomponent Entry to Polysubstituted 2-Aminopyrroles
- Palladium-Catalyzed Synthesis of Arylgermanium Compounds
- Synthesis of 1-Monosubstituted 1,2,3-Triazoles
- Continuous-Flow Synthesis of Chiral 1,2-Diamino Derivatives
- New Synthesis of Azulene
- A Synthesis of S,S-DICHED Catalyst for Matteson Homologations
- Novel Oxazole-Containing Amino Acids
- B-Ring Contraction in Steroids via Benzilic Acid Rearrangement
- Photoredox Synthesis of Arylhydroxylamines
- Unsymmetrical Biheteroaryls via Suzuki–Miyaura Cross-Couplings Using an Air-Stable Pre-Catalyst
- Mechanistic Insight on the Bromocycloetherification of Alkenes
- Synthesis of Arylalkynes from Diaryl Sulfoxides
- SYNLETT Editorial Board Welcomes New Members
- New Heptitol Derivatives as Potential Antibacterials
- New Entry to Cyclopentyl Aryl Ketones via Photoredox Catalysis
- Iodide-Catalyzed Carbonylation–Benzylation of Benzyl Chlorides
- Synthesis of Functionalized Rubicenes
- Pd-Catalyzed Synthesis of ortho-Fluorodiarylmethanes
- Novel Entry to Tetraarylmethanes
- Synthesis of N-Arylsulfonamides
- Monofluoro Aryl Acetates via Copper Catalysis
- Enaminones via Palladium-Catalyzed Four-Component Carbonylation
- Trifluoromethylation of Highly Functionalized Heteroarenes: Flow to the Rescue
- Novel Synthesis of Aryl Cyclopropylketones
- Total Synthesis of Lagerstannin C
- New Synthetic Access to Ethers
- Stereoselective Cyclopropanation of (–)-Levoglucosenone Derivatives
- Microwave-Promoted Synthesis of 4-Arylpyrimidines in Water
- Protein Synthesis and Crystallization of Bowman–Birk Protease Inhibitors
- Improved Fmoc Deprotection Methods for the Synthesis of Thioamide-Containing Peptides and Proteins
- Synthesis of 3,5,7-Trisubstituted Indoles
- Rhodium(III)-Catalyzed Sulfonamidation of Azoxybenzenes
- Synthesis and Properties of 2-Oxa-6-azaspiro[3.3]heptane Sulfonate Salts
- Metal-Free Primary Amination of Potassium Aryltrifluoroborates and Phenylboronic Acids
- Synthesis of a Ubiquitinated Histone Mimic Bearing a New Thioether Linkage
- Organocatalytic Synthesis of non-Racemic Oxazolines from Isocyanoacetate and α-Keto Esters
- Catalytic Asymmetric α-Hydroxylation of 3-Substituted Oxindoles with Hydrogen Peroxide
- Synthesis of Benzo[e]azolo[1,3]oxazines
- Preparation of 3-Aminoimidazo[1,2-a]pyrazines
- [3+2] Cycloaddition of Azomethine Ylides
- Synthesis of N,O-Nucleosides via Ene Reaction
- Bunte Salts as Thiolating Reagents for Alkenes
- Synthesis of Fused Naphthobenzofurans
- New Entry to Tetrahydropyrazolopyrazolones via [3+2] Cycloaddition
- Enantiocontrolled Synthesis of Non-racemic γ-Acetoxyallylboronates
- Asymmetric Aldol Reactions with a Dual Catalyst System
- Multistep Continuous-Flow Synthesis of (–)-Oseltamivir
- Synthesis of the Siderophore Erythrochelin
- New Parallel Synthesis of Di(hetero)arylamides
- Augmented Reality as an Enabling Tool in Organic Chemistry
- Lanthanum-Catalyzed Olefination of Benzylamines with 2-Methylquinoline via Tandem Oxidation/Benzylidene Addition
- Efficient Access to the Structural Core of Annonaceous Acetogenins
- Synthesis of α-Arylglycines and Other α-Amino Acid Derivatives
- New Synthesis of Morpholines and Benzoxazines
- Synthesis and Structural revision of a γ-Lactone Polyketide of Fungal Origin
- 2-Alkynyl-1,4-cyclohexadienes via a Diels–Alder Reaction
- Aryltrimethylgermanes for the Arylation of Amines and Amides
- Samarium(II)-Promoted Synthesis of 2-Azabicycles
- First Total Synthesis of Dermocanarin 2
- Synthesis of Enantiopure tert-Butylmethylphosphine–Boranes
- Total Synthesis of δ-Sanshool and Analogues
- Novel Entry to Peptides Incorporating Tryptophan and Analogues
- Photoredox Catalysis for a Novel Access to Pentafluorosulfanyl Compounds
- Novel Substrates for Desymmetrization Processes
- Enantiopure Monomethylated L-Arginine and L-Ornithine
- Iodo- and Chloroamination of Enecarbamates
- Enantioselective N-Functionalization of Pyrroles
- Novel Fluorescently Labeled Amino Acids
- Synthesis of Enantiomerically Pure β-Methoxytyrosine
- Novel Route to Aromatic Hydrazines via Cu-Catalyzed Addition of Arylboronic Esters to Azodicarboxylates
- Novel Synthesis of Orthogonally Protected Diazaspiro[3.4]octane Analogues
- Trityl Group Deprotection from Tetrazoles
- Synthesis of Cyclotribenzoin
- Synthesis of New Chiral Diaryliodonium Salts
- Synthesis and Analysis of Macrocyclic Peptides with 310-Helical Structure
- Total Synthesis of (+)-Clavulatriene A
- Biologically Important Phosphotriesters by Organocatalysis
- New Potential Organic Semiconductors